4-Methylamino antipyrine
CAS No. 519-98-2
4-Methylamino antipyrine ( —— )
Catalog No. M26030 CAS No. 519-98-2
4-Methylamino antipyrine is an active metabolite of Metamizole. Metamizole is a pyrazolone non-steroidal anti-inflammatory drug (NSAID) and inhibits COX.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
10MG | 35 | In Stock |
|
25MG | 76 | In Stock |
|
50MG | 113 | In Stock |
|
100MG | 176 | In Stock |
|
200MG | 268 | In Stock |
|
500MG | 446 | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
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Product Name4-Methylamino antipyrine
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NoteResearch use only, not for human use.
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Brief Description4-Methylamino antipyrine is an active metabolite of Metamizole. Metamizole is a pyrazolone non-steroidal anti-inflammatory drug (NSAID) and inhibits COX.
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Description4-Methylamino antipyrine is an active metabolite of Metamizole. Metamizole is a pyrazolone non-steroidal anti-inflammatory drug (NSAID) and inhibits COX. 4-Methylamino antipyrine has analgesic, antipyretic, and relatively weak anti-inflammatory properties.(In Vitro):At room temperature and in an atmosphere with oxygen, Metamizole is spontaneously, nonenzymatically converted to 4-Methylamino antipyrine. Subsequently, the N-methyl side chain of 4-Methylamino antipyrine is oxidized to yield 4-formylaminoantipyrine, which is further converted to 4-aminoantipyrine .(In Vivo):Eight healthy male piglets are administered Metamizole (100 mg/kg) intramuscularly. 4-Methylamino antipyrine plasma concentrations are quantitatively detectable from 0.25 to 48 h. The average maximum concentration of 4-Methylamino antipyrine is 47.59 mg/mL. The average half-lives is 8.57 h for 4-Methylamino antipyrine .
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetCOX
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RecptorCRAC channel
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Research Area——
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Indication——
Chemical Information
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CAS Number519-98-2
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Formula Weight217.3
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Molecular FormulaC12H15N3O
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Purity>98% (HPLC)
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Solubility——
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SMILESCNc1c(C)n(C)n(-c2ccccc2)c1=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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